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Bioanalytical Services
Leading LC-MS/MS-laboratory in Europe with more than
100 validated LC-MS/MS-assays
Largest worldwide experience in LC-MS/MS of antiinfectives including modern antiretroviral compounds
LC-UV/fluorescence assays:
More than 300 validated assays
Bioavailability and Pharmacokinetic Studies
Bioequivalence
Drug-drug interaction,
Food-drug interaction
Dose-proportionality studies
Quality Service
Pharmacodynamic studies
Studies in Eastern Europe
Full study service (consulting, report writing), publications
Pharmacokinetic modeling using Kinetica, SIPHAR, P-Pharm, NONLIN, TOPFIT, NONMEM
Statistical services using SAS
PK-PD modeling
Bioequivalence services
In vitro - in vivo correlation (Level A-C acc. to USP XVIII)
In vivo dissolution studies
Special studies
Drug penetration into uninflamed or inflamed CSF (new drug entities) in man (only therapeutically relevant agents in these patients).
Phototoxicity studies in man.
Model of drug distribution by analysis of body fluids such as saliva, sweat, tears, nasal secretion, prostatic fluid.
In vitro - in vivo protein and cell binding studies.
Liver: microsomal perfusion, hepatocyte work.
Studies on gastrointestinal site of absorption by local application of drug solutions and/or tablets with predependent dissolving coatings.
Probe-studies using newly developed drug cocktails to assess drug absorption, metabolism and elimination simultaneously
Tissue Penetration Studies:
Microdialysis
Blister fluid
Sputum
Body fluids: salvia, sweat, tears; nasal secretions, prostatic fluid (integrated body fluid model)
Single cell concentration measurement
Prostatic fluid and sperm
CSF
Peritoneal fluid, bronchial lavage
Feces
Saliva
Tissues: prostatic, lung, bronchial, bone, muscle, fat and virtually any other tissue in humans.
Special populations:
obese subjects
breast-feeding mothers
post-menopausal women
women on oral contraceptives
hepatic insufficiency patients
poor metabolizer studies
intestinal elimination
studies with charcoal model + feces in humans
cystic fibrosis patients
middle aged subjects
HIV-positive patients
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